Ukuhlukahluka kokuthambekela | N / a |
Cas cha | 71963-77-4 |
Uhlobo lwamakhemikhali | C16h26o5 |
Isisindo molecular | 298.37 |
Ama-eInec no. | I-663-549-0 |
Iphuzu elincibilikayo | 86-88 ° C |
Iphuzu elibilayo | 359.79 ° C (isilinganiso esibi) |
Ukujikeleza okuthile | D19.5 + 171 ° (C = 2.59inCH3) |
Incekusana | I-1.0733 (isilinganiso esinzima) |
Inkomba ye-refraction | 1.6200 (ukulinganisa) |
Izimo Zokugcina | Igumbi lekamelo |
Ubuhlakaniselo | DMSOSYMG / ML |
Ukubonakala | Impushana |
Amanyanjana | I-Arteremerum / artemtherin / dihydroartemisinmethylether |
Ubuhlakaniselo | Incibilika emanzini |
Izigaba | Isitshalo esikhishwe, isengezo, ukunakekelwa kwempilo |
Izinja | Anti-malarial |
Inzalo yi-sactone ye-sactone etholakala ezimpandeni zeI-Artemisia Annua, ojwayele owaziwa ngokuthi umhlonyane omnandi. Kuyisidakamizwa esinamandla esingonakaliso esisetshenziselwa ukwelapha nokuvimbela umalaleveva. I-Artemisinin, isandulelo sezinstrumlezwe, sakhishwa okokuqala esitshalweni ngawo-1970, futhi ukutholwa kwaso kwathola umcwaningi waseChina uTu umklomelo kaNobel kwezokwelapha ngo-2015.
Sekusebenza ngobuhlungu ngokubhubhisa ama-parasites abhekele umala umalaleveva. Umalaleveva kubangelwa yi-protozoan parasite ebizwa ngePlasmodium, edluliselwa kubantu ngokuluma komiyane wabesifazane abanegciwane. Lapho nje umgcini womuntu, ama-parasites aphindaphindeka kakhulu esibindini kanye namangqamuzana abomvu egazi, abangela umkhuhlane, amabala, nezinye izimpawu ezinjengemfuli. Uma kushiywe kungalashwa, umalaleveva angabulala.
Izinkundla zemidlalo zisebenza kakhulu ekulweni nezinkinga ezingazweli emishangubeni zePlasmodium Falciparum, okuthi yinqwaba yokufa kwabantu abahlobene nemalaleveva emhlabeni jikelele. Kuyaphumelela futhi ngokumelene nezinye izinhlobo zama-plasmodium parasites abangela umalaleveva. Sekuvamiswe ukuhanjiswa ngokuhlanganiswa nezinye izidakamizwa, njenge-lumefantrine, ukunciphisa ingozi yokumelana nezidakamizwa.
Ngaphandle kokusetshenziswa kwayo njengesidakamizwa esingonakalisi, sekutholakele futhi kube nezinye izakhiwo zokwelapha. Ucwaningo selukhombisile ukuthi linokulwa nokuvuvukala, anti-isimila, kanye nemisebenzi elwa namagciwane. Kusetshenziselwe ukwelapha isifo samathambo, i-lupus, nezinye izifo ze-autoimmune. Kubuye kwaphenywa ngamathuba alo okuphamba i-Covid-19, yize kudingeka ucwaningo oluningi ukuze kuqinisekiswe ukusebenza kwalo.
Izingqinamba ngokuvamile ziphephile futhi zibekezelelwa kahle lapho zisetshenziswa njengoba kuqondiswa. Kodwa-ke, njengazo zonke izidakamizwa, kungadala imiphumela emibi. Imiphumela emibi evame kakhulu yemizwa yezingcingo ifaka phakathi isicanucanu, ukugabha, isiyezi, kanye nekhanda. Ezimweni ezingavamile, kungadala ukusabela okubi kakhulu, njengezinhliziyo ze-paltiations, kubanjwa, kanye nomonakalo wesibindi.
Ekuphetheni, ubuthi yinhloso umuthi onamandla aphikisayo oguqule ukwelashwa umalaleveva nokuvimbela. Ukutholwa kwayo kusindise izimpilo ezingenakubalwa futhi kwathola ukuqashelwa komphakathi wesayensi. Enye indawo yayo yokwelapha yenza kube ngumuntu othembisayo ekwelapheni ezinye izifo. Yize kungadala imiphumela emibi, izinzuzo zawo zidlula kude kakhulu izingozi zayo lapho zisetshenziswa ngaphansi kokugadwa kwezokwelashwa.
Amafomu we-DOSAge asetshenziswa kakhulu afaka amaphilisi, amaphilisi nemijovo. Izinhlobo zezidakamizwa ziyizidakamizwa ezilwa namagciwane, futhi ingxenye enkulu yobuhlungu. Umlingiswa onesibopho sezibhebhethezi kwakukhona amaphilisi amhlophe. Isimo se-ardereneature capsule yi-capsule, okuqukethwe okungumpuphu omhlophe; Umlingiswa wezidakamizwa we-tortenereaseatjolo awunamibala ukukhanyisa uwoyela ophuzi - njengoketshezi.
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